Efficient C3-alkylsulfenylation of indoles under mild conditions using Lewis acid-activated 8-quinolinethiosulfonates
نویسندگان
چکیده
The activation of 8-quinolinethiosulfonates by zinc chloride promotes the usually difficult to achieve C3-alkylsulfenylation indoles at room temperature under aerobic conditions. This strategy is compatible with substrates containing various functional groups.
منابع مشابه
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ژورنال
عنوان ژورنال: Tetrahedron Letters
سال: 2021
ISSN: ['0040-4039', '1873-3581']
DOI: https://doi.org/10.1016/j.tetlet.2020.152748